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Tocainide hydrochloride
CAS No. 71395-14-7
Tocainide hydrochloride ( 2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride )
Catalog No. M24724 CAS No. 71395-14-7
Tocainide hydrochloride is a sodium channel blocker. It blocks the sodium channels in the pain-producing foci in the nerve membranes.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 500MG | 1796 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTocainide hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionTocainide hydrochloride is a sodium channel blocker. It blocks the sodium channels in the pain-producing foci in the nerve membranes.
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DescriptionTocainide hydrochloride is a sodium channel blocker. It blocks the sodium channels in the pain-producing foci in the nerve membranes.
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In Vitro——
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In VivoTocainide (100 mg/kg) effectively suppresses ventricular ectopic activity in unanesthetized dogswith coronary occlusion. Termination of tocainide infusion in both digitalis toxicity and coronary occlusion models results in prompt return of ventricular ectopic activity.
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Synonyms2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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RecptorSodium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number71395-14-7
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Formula Weight228.72
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Molecular FormulaC11H17ClN2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (546.52 mM)
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SMILESCl.CC(N)C(=O)Nc1c(C)cccc1C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Alpert JS, et al. Chemistry, pharmacology, antiarrhythmic efficacy and adverse effects of tocainide hydrochloride, an orally active structural analog of lidocaine. Pharmacotherapy. 1983 Nov-Dec;3(6):316-23.
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